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本书分为理论和实验两大部分,理论部分共十六章,实验部分有六个实验。重点叙述了化学药物的结构、性质、稳定性及构效关系等,简单叙述了各大类药物的发展过程、最新进展及体内代谢,对药物的合成也作了适当的介绍。